SCHEMBL8319085

SCHEMBL8319085

CS(=O)(=O)c1ncc2ncnc(Nc3ccc(N)c([N+](=O)[O-])c3)c2n1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.44
ABCG2 Q9UNQ0 3/20 0.42
FFAR4 Q5NUL3 1/20 0.39
DYRK1A Q13627 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA13 Q8N1Q1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318233 0.88 EGFR (0.47) EGFRABCG2CA1CA2CA7
SCHEMBL6994362 0.84 ABCG2 (0.56) EGFRABCG2
SCHEMBL8317837 0.83 EGFR (0.45) EGFRABCG2DYRK1ADYRK1B
SCHEMBL8314779 0.82 EGFR (0.45) EGFR
SCHEMBL6997375 0.78 EGFR (0.47) EGFR
SCHEMBL8317145 0.78 EGFR (0.49) EGFRDYRK1ADYRK1B
SCHEMBL6991028 0.77 GSK3A (0.55) EGFRABCG2
SCHEMBL6991037 0.77 GSK3A (0.55) EGFRABCG2
SCHEMBL6995080 0.76 BRAF (0.49)
SCHEMBL6417047 0.76 EGFR (0.66) EGFRABCG2DYRK1ADYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed