SCHEMBL8314899

SCHEMBL8314899

O=C(O)C1=CC(CF)(CF)Oc2ccc(Cl)cc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
TP53 P04637 2/20 0.36
NOTUM Q6P988 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
AKR1B1 P15121 1/20 0.34
HCAR2 Q8TDS4 1/20 0.33
TSHR P16473 2/20 0.33
CASP1 P29466 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HPGD P15428 1/20 0.32
KDM4E B2RXH2 2/20 0.32
MCL1 Q07820 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
GPR35 Q9HC97 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TTR P02766 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313550 0.84 ALDH1A1 (0.35) ALDH1A1TP53AKR1B1TSHRKDM4E
SCHEMBL8316159 0.83 AKR1B1 (0.32) PTGS1PTGS2AKR1B1
SCHEMBL8313695 0.78 KDM4E (0.34) ALDH1A1TP53KDM4EL3MBTL1ALPG
SCHEMBL8316624 0.76 KDM4E (0.30) KDM4E
SCHEMBL7093857 0.68 CHRM1 (0.33) PTGS1PTGS2PTGDR2
SCHEMBL6269700 0.67 ALDH1A1 (0.36) ALDH1A1CA1CA2TSHRCASP1
SCHEMBL8574539 0.62 SMN1; SMN2 (0.57) ALDH1A1TP53CA1CA2TSHR
SCHEMBL27675905 0.62 ALDH1A1 (0.57) ALDH1A1TP53NOTUMCA1CA2
SCHEMBL2829838 0.62 LMNA (0.59) ALDH1A1TP53CA2PTGS1PTGS2
SCHEMBL2433995 0.61 PPOX (0.41) ALDH1A1HPGDKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632033-B1 NOVEL BENZOPYRAN DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 1999-04-07 EP disclosed
US-5646308-A POTASSIUM CHANNEL ACTIVATORS USED AS ANTIASTHMATICS, ANTIEPILEPTICS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1997-07-08 US disclosed
EP-0632033-A1 NOVEL BENZOPYRAN DERIVATIVE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1995-01-04 EP disclosed