SCHEMBL8314119

SCHEMBL8314119

CC1(C)COc2ccc(-c3ccccc3)cc2C(O)(c2ccccn2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.38
TMEM97 Q5BJF2 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
HTR7 P34969 1/20 0.38
HTR1A P08908 1/20 0.37
SLC6A2 P23975 1/20 0.36
BACE1 P56817 5/20 0.35
CTSD P07339 2/20 0.34
NOTUM Q6P988 2/20 0.34
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316835 0.86 SLC6A2 (0.39) HTR2BSIGMAR1HTR1ASLC6A2NPC1
SCHEMBL8311266 0.86 SLC6A2 (0.37) SLC6A2BACE1PDK2
SCHEMBL8311974 0.85 BACE1 (0.37) SLC6A2BACE1MAPTKMT2ASMN1; SMN2
SCHEMBL8313637 0.85 SLC6A2 (0.36) SLC6A2BACE1NPC1RAB9AKMT2A
SCHEMBL8310708 0.84 SLC6A2 (0.40) HTR1ASLC6A2KMT2ASMN1; SMN2PDK2
SCHEMBL8314935 0.83 SCN9A (0.38) HTR2BTMEM97SIGMAR1HTR7HTR1A
SCHEMBL8313905 0.83 PDK2 (0.35) SLC6A2BACE1RAB9AKMT2APDK2
SCHEMBL8313766 0.83 PDK2 (0.35) SLC6A2PDK2
SCHEMBL8314864 0.83 SLC6A2 (0.37) SLC6A2NPC1RAB9ASMN1; SMN2
SCHEMBL8313558 0.82 SLC6A2 (0.38) SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed