SCHEMBL8313637

SCHEMBL8313637

CC1(C)COc2ccc(Cl)cc2C(O)(c2ccccn2)C1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.36
MAP3K14 Q99558 1/20 0.35
SLC6A9 P48067 4/20 0.35
NR3C1 P04150 1/20 0.32
RAB9A P51151 2/20 0.32
NPC1 O15118 1/20 0.32
KMT2A Q03164 1/20 0.32
BACE1 P56817 2/20 0.32
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313558 0.88 SLC6A2 (0.38) SLC6A2MAP3K14SLC6A9NR3C1
SCHEMBL8316835 0.87 SLC6A2 (0.39) SLC6A2NR3C1RAB9ANPC1
SCHEMBL8311266 0.87 SLC6A2 (0.37) SLC6A2BACE1
SCHEMBL8311974 0.86 BACE1 (0.37) SLC6A2KMT2ABACE1
SCHEMBL8310708 0.85 SLC6A2 (0.40) SLC6A2NR3C1KMT2A
SCHEMBL8314119 0.85 HTR2B (0.38) SLC6A2RAB9ANPC1KMT2ABACE1
SCHEMBL8313766 0.84 PDK2 (0.35) SLC6A2
SCHEMBL8315996 0.84 SLC6A2 (0.35) SLC6A2NR3C1BACE1
SCHEMBL8314935 0.84 SCN9A (0.38) SLC6A2RAB9ANPC1KMT2ABACE1
SCHEMBL8313905 0.84 PDK2 (0.35) SLC6A2NR3C1RAB9AKMT2ABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed