SCHEMBL8315262

SCHEMBL8315262

COc1cc(/C=C/c2nc3c(s2)NCCCC3)cc(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
CYP1A1 P04798 8/20 0.41
CYP1B1 Q16678 8/20 0.41
CYP1A2 P05177 5/20 0.40
NQO2 P16083 6/20 0.37
ABL1 P00519 3/20 0.37
BCR P11274 3/20 0.37
TTR P02766 3/20 0.37
ESR1 P03372 2/20 0.37
ABCB1 P08183 2/20 0.37
ALOX5 P09917 2/20 0.37
CYP19A1 P11511 2/20 0.37
PTGS2 P35354 2/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
AHR P35869 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315265 1.00 PARP1 (0.46) PARP1CYP1A1CYP1B1CYP1A2NQO2
SCHEMBL8317005 0.88 KDM4E (0.42) CYP1A1CYP1B1CYP1A2NQO2ABL1
SCHEMBL8317001 0.88 KDM4E (0.42) CYP1A1CYP1B1CYP1A2NQO2ABL1
Hydrochloric Acid SCHEMBL8311790 0.88 RELA (0.42) CYP1A1CYP1B1CYP1A2NQO2CYP19A1
Hydrochloric Acid SCHEMBL8311789 0.88 RELA (0.42) CYP1A1CYP1B1CYP1A2NQO2CYP19A1
SCHEMBL8314240 0.86 KDM4E (0.45) CYP1A1CYP1B1CYP1A2NQO2CYP19A1
SCHEMBL8314245 0.86 KDM4E (0.45) CYP1A1CYP1B1CYP1A2NQO2CYP19A1
Hydrochloric Acid SCHEMBL8459129 0.85 KDM4E (0.44) CYP1A1CYP1B1CYP1A2TUBB4ATUBB
Hydrochloric Acid SCHEMBL8459126 0.85 KDM4E (0.44) CYP1A1CYP1B1CYP1A2TUBB4ATUBB
SCHEMBL9694219 0.82 ALDH1A1 (0.45) CYP1A1CYP1B1CYP1A2NQO2TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0351856-B1 Thiazolo[5,4-b]azepine compounds TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-09-15 EP disclosed
US-4956360-A LIPOPEROXIDE INHIBITORS, ENZYME INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-09-11 US disclosed