SCHEMBL8315434

SCHEMBL8315434

c1ccc(CN2CCC(C3CCN(Cc4ccccc4)CC3)CC2)cc1

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.71
SIGMAR1 Q99720 4/20 0.71
CCR3 P51677 1/20 0.69
DRD2 P14416 2/20 0.65
DRD4 P21917 2/20 0.65
DRD3 P35462 2/20 0.65
BACE1 P56817 2/20 0.62
BCHE P06276 1/20 0.62
ALDH1A1 P00352 1/20 0.59
CXCR4 P61073 1/20 0.59
HTR2A P28223 1/20 0.59
MC4R P32245 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7319631 0.92 ACHE (0.62) ACHESIGMAR1CCR3DRD2DRD4
SCHEMBL13432184 0.91 MC4R (0.70) ACHESIGMAR1CCR3DRD2DRD4
SCHEMBL3352682 0.89 SIGMAR1 (0.68) ACHESIGMAR1CCR3DRD2DRD4
SCHEMBL1232375 0.88 ACHE (0.67) ACHESIGMAR1CCR3DRD2DRD4
Hydrochloric Acid SCHEMBL20607541 0.88 SIGMAR1 (0.66) ACHESIGMAR1CCR3DRD2DRD4
SCHEMBL22728510 0.87 ACHE (0.61) ACHESIGMAR1CCR3DRD2DRD4
SCHEMBL13154555 0.86 ACHE (0.56) ACHESIGMAR1CCR3DRD2DRD4
Hydrochloric Acid SCHEMBL28439633 0.86 ACHE (0.65) ACHESIGMAR1CCR3DRD2DRD4
SCHEMBL2087027 0.85 ACHE (0.59) ACHESIGMAR1CCR3DRD2DRD4
SCHEMBL6182247 0.85 HRH3 (0.59) ACHESIGMAR1CCR3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004066960-A2 COMBINATION OF H1, H3 AND H4 RECEPTOR ANTAGONISTS FOR TREATMENT OF ALLERGIC AND NON-ALLERGIC PULMONARY INFLAMMATION, CONGESTION AND ALLERGIC RHINITIS SCHERING CORPORATION (US) 2004-08-12 WO disclosed