SCHEMBL8315540

SCHEMBL8315540

O=C(Cc1ccccc1)Nc1ccc(C(=O)N2CCc3cccn3-c3ccccc32)cc1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.48
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
NR4A1 P22736 1/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KMT2A Q03164 3/20 0.46
NPY2R P49146 1/20 0.45
EPHX2 P34913 1/20 0.45
NAMPT P43490 1/20 0.44
KCNQ2 O43526 1/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416297 0.89 HSD11B1 (0.47) HSD11B1KDM4EALDH1A1MAPTNR4A1
SCHEMBL8312803 0.86 AVPR2 (0.49) KMT2AMEN1
SCHEMBL8318866 0.86 KCNJ5 (0.47) NAMPTKCNQ2
SCHEMBL7332706 0.83 AVPR2 (0.47) KMT2ANAMPTMEN1
SCHEMBL8558667 0.79 NAMPT (0.54) HSD11B1KDM4EALDH1A1MAPTNR4A1
SCHEMBL8315722 0.78 AVPR1A (0.64)
SCHEMBL8314568 0.78 AVPR1A (0.58) HSD11B1
SCHEMBL8314325 0.78 AVPR1A (0.52) KMT2AMEN1
SCHEMBL8315401 0.78 AVPR1A (0.51)
SCHEMBL7349542 0.78 AVPR1A (0.65) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed