SCHEMBL8315609

SCHEMBL8315609

O=CNCC(CCO)(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH1B P00325 1/20 0.40
ADH1C P00326 1/20 0.40
ADH1A P07327 1/20 0.40
ADH7 P40394 1/20 0.40
ALDH1A1 P00352 2/20 0.35
CHRM2 P08172 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
TSHR P16473 1/20 0.32
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
CYP2C19 P33261 2/20 0.31
CCR1 P32246 2/20 0.31
CCR3 P51677 2/20 0.31
KCNN4 O15554 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7823386 0.90 ADH1B (0.38) ADH1BADH1CADH1AADH7ALDH1A1
SCHEMBL7822809 0.89 CCR3 (0.37) ADH1BADH1CADH1AADH7ALDH1A1
SCHEMBL8893131 0.85 CCR1 (0.35) ADH1BADH1CADH1AADH7ALDH1A1
SCHEMBL7816549 0.82 CCR3 (0.45) MEN1KMT2ACCR1CCR3LMNA
SCHEMBL7817328 0.80 ADH1B (0.38) ADH1BADH1CADH1AADH7ALDH1A1
SCHEMBL7824381 0.79 KIF11 (0.43) ALDH1A1MEN1KMT2ACCR1CCR3
SCHEMBL7827162 0.79 ADH1B (0.37) ADH1BADH1CADH1AADH7ALDH1A1
SCHEMBL29097001 0.77 TDP1 (0.40) ALDH1A1CHRM2CHRM1CHRM3TSHR
SCHEMBL7468423 0.76 LMNA (0.46) ALDH1A1CHRM2CHRM1CHRM3CHRM4
SCHEMBL8892088 0.76 KIF11 (0.35) ADH1BADH1CADH1AADH7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0679642-B1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-11-10 EP disclosed
US-5654296-A HORMONE INHIBITOR; NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-08-05 US disclosed
US-5607939-A CALCIUM ANTAGONIST, GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONIST AND MONOAMINEU UPTAKE INHIBITORS FOR CENTRAL NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-04 US disclosed
EP-0679642-A1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-02 EP disclosed