SCHEMBL8316488

SCHEMBL8316488

COc1cc2c(cc1OC)C(c1ccccn1)=CC(C)(C)CO2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.40
POLB P06746 2/20 0.38
KDM4E B2RXH2 5/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
NPC1 O15118 3/20 0.38
TP53 P04637 2/20 0.38
RAB9A P51151 2/20 0.38
HSD17B10 Q99714 2/20 0.38
GAA P10253 1/20 0.38
PKM P14618 1/20 0.38
PDE4A P27815 1/20 0.36
MAPT P10636 4/20 0.36
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.35
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313611 0.84 NPC1 (0.41) KDM4ESMN1; SMN2NPC1RAB9AGAA
SCHEMBL8311427 0.82 SCN9A (0.35) POLBKDM4ERAB9AALDH1A1LMNA
SCHEMBL8316296 0.82 CCR1 (0.35) POLBKDM4ESMN1; SMN2NPC1TP53
SCHEMBL8875966 0.81 NPY5R (0.34) POLBKDM4ESMN1; SMN2LMNAHTT
SCHEMBL8316184 0.80 KDM4E (0.37) POLBKDM4ESMN1; SMN2NPC1TP53
SCHEMBL8315486 0.80 NPC1 (0.39) POLBKDM4ESMN1; SMN2NPC1TP53
SCHEMBL8315309 0.79 ADRA1A (0.38) POLBKDM4ESMN1; SMN2NPC1TP53
SCHEMBL8312863 0.79 MAPT (0.39) KDM4ESMN1; SMN2NPC1TP53RAB9A
SCHEMBL8315585 0.79 ADRA1A (0.40) POLBKDM4ESMN1; SMN2NPC1TP53
SCHEMBL8314584 0.79 FABP6 (0.37) RAB9AMAPTGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed