SCHEMBL8315796

SCHEMBL8315796

O=CNCC(CCN1CCN(c2ccc(F)cc2)CC1)(c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.48
REV1 Q9UBZ9 1/20 0.47
KCNA3 P22001 1/20 0.47
LMNA P02545 2/20 0.46
GAA P10253 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
DRD2 P14416 1/20 0.44
HTR2A P28223 1/20 0.44
HRH1 P35367 1/20 0.44
DRD3 P35462 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CHRM4 P08173 1/20 0.42
CHRM3 P20309 1/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8310440 0.99 HTR1A (0.47) HTR1AREV1KCNA3LMNAGAA
SCHEMBL7470176 0.93 CHRM4 (0.48) HTR1ADRD2HTR2AHRH1DRD3
SCHEMBL7458791 0.92 DRD2 (0.47) HTR1ADRD2HTR2AHRH1DRD3
Hydrochloric Acid SCHEMBL7459516 0.92 CHRM4 (0.50) HTR1ADRD2HTR2AHRH1DRD3
Hydrochloric Acid SCHEMBL7464721 0.91 CHRM4 (0.46) HTR1ADRD2HTR2AHRH1DRD3
SCHEMBL7462282 0.88 DRD2 (0.49) HTR1ADRD2HTR2AHRH1DRD3
Hydrochloric Acid SCHEMBL7459710 0.87 DRD2 (0.49) HTR1ADRD2HTR2AHRH1DRD3
SCHEMBL8313258 0.85 CHRM4 (0.56) HTR1AKCNA3DRD2HTR2AHRH1
SCHEMBL7464684 0.84 DRD2 (0.49) HTR1ADRD2HTR2AHRH1DRD3
SCHEMBL7471015 0.83 DRD2 (0.53) HTR1ALMNADRD2HTR2AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0679642-B1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-11-10 EP disclosed
US-5654296-A HORMONE INHIBITOR; NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-08-05 US disclosed
US-5607939-A CALCIUM ANTAGONIST, GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONIST AND MONOAMINEU UPTAKE INHIBITORS FOR CENTRAL NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-04 US disclosed
EP-0679642-A1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-02 EP disclosed