SCHEMBL8315892

SCHEMBL8315892

CC(=O)NC(Cc1csc2ccccc12)(C(=O)O)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.48
CYP2A6 P11509 2/20 0.47
TAAR1 Q96RJ0 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
TP53 P04637 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
POLB P06746 1/20 0.44
FAAH O00519 1/20 0.44
MAPT P10636 1/20 0.43
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
HDAC6 Q9UBN7 2/20 0.41
TACR1 P25103 1/20 0.41
HDAC1 Q13547 1/20 0.41
MTNR1A P48039 1/20 0.41
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8486768 0.79 CYP2A6 (0.59) CYP2A6TAAR1SMN1; SMN2TP53RXFP1
SCHEMBL10950583 0.79 CYP2A6 (0.54) PKMCYP2A6TAAR1SMN1; SMN2TP53
SCHEMBL2534944 0.77 CYP2A6 (0.53) PKMCYP2A6TAAR1SMN1; SMN2TP53
SCHEMBL9265036 0.75 TACR1 (0.55) PKMCYP2A6TAAR1SMN1; SMN2TP53
SCHEMBL21274459 0.73 SMN1; SMN2 (0.61) CYP2A6TAAR1SMN1; SMN2TP53RXFP1
SCHEMBL4659729 0.73 CYP2A6 (0.48) PKMCYP2A6TAAR1SMN1; SMN2TP53
SCHEMBL28168069 0.73 ALDH1A1 (0.67) SMN1; SMN2MAPT
SCHEMBL1686166 0.73 ALDH1A1 (0.44) MAPTMTNR1A
Acetic Acid SCHEMBL7564503 0.72 CYP2A6 (0.58) PKMCYP2A6TAAR1SMN1; SMN2TP53
SCHEMBL760833 0.71 MTNR1A (0.67) PKMCYP2A6TAAR1SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635508-B1 TETRAHYDROPYRIDINE DERIVATIVE HAVING SUBSTITUENTS ON THREE RINGS ASAHI CHEMICAL IND (JP) 1999-10-06 EP disclosed
US-5621103-A 3-(SUBSTITUTED METHYLAMINOCARBONYL)-1,2,3,4-TETRAHYDRO-(1)BENZOTHIENO(2,3-C) PYRIDINES; ANXIOLYTIC AGENTS; LEARNING ENHANCEMENT ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1997-04-15 US disclosed
EP-0635508-A1 TETRAHYDROPYRIDINE DERIVATIVE HAVING SUBSTITUENTS ON THREE RINGS Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-01-25 EP disclosed
EP-0386258-A1 TETRAHYDROPYRIDINE DERIVATIVES Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1990-09-12 EP disclosed