SCHEMBL8316487

SCHEMBL8316487

O=C(Nc1ccc(C(=O)N2CCc3cccn3-c3ccccc32)c(Cl)c1)c1ccccc1OC(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 11/20 0.49
AVPR2 P30518 11/20 0.49
PNLIP P16233 1/20 0.49
OXTR P30559 1/20 0.46
RXFP1 Q9HBX9 1/20 0.45
KCNK3 O14649 3/20 0.44
KCNK9 Q9NPC2 3/20 0.44
F2R P25116 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316224 0.87 AVPR2 (0.44) AVPR1AAVPR2OXTRRXFP1
SCHEMBL8313809 0.84 AVPR2 (0.69) AVPR1AAVPR2OXTR
SCHEMBL7333870 0.84 AVPR2 (0.64) AVPR1AAVPR2OXTR
SCHEMBL7334076 0.82 AVPR2 (0.68) AVPR1AAVPR2OXTR
SCHEMBL7341288 0.82 AVPR2 (0.68) AVPR1AAVPR2OXTR
SCHEMBL7415555 0.78 AVPR2 (0.49) AVPR1AAVPR2
SCHEMBL6989072 0.77 AVPR1A (0.55) AVPR1AAVPR2PNLIPKCNK3KCNK9
SCHEMBL8318107 0.76 AVPR2 (0.65) AVPR1AAVPR2
SCHEMBL8314568 0.76 AVPR1A (0.58) AVPR1AAVPR2
SCHEMBL8317555 0.75 AVPR2 (0.54) AVPR1AAVPR2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed