SCHEMBL8313611

SCHEMBL8313611

COc1ccc2c(c1)C(c1ccccn1)=CC(C)(C)CO2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
ALOX12 P18054 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
NPY5R Q15761 1/20 0.40
RUNX1 Q01196 1/20 0.39
CYP19A1 P11511 2/20 0.39
PKM P14618 2/20 0.38
HTR2B P41595 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
GRM5 P41594 1/20 0.38
HTR7 P34969 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
TGFBR1 P36897 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315603 0.86 CBFB (0.42) RUNX1GRM5BACE1SCN9ACTSD
SCHEMBL8316488 0.84 PDE10A (0.40) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8315486 0.84 NPC1 (0.39) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8315585 0.83 ADRA1A (0.40) NPC1RAB9ASMN1; SMN2KDM4EMAPT
SCHEMBL8312863 0.83 MAPT (0.39) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8314584 0.83 FABP6 (0.37) RAB9AMAPTNPY5RCYP19A1GRM5
SCHEMBL8316184 0.82 KDM4E (0.37) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8310381 0.82 HTR2B (0.40) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8312053 0.81 TGFBR1 (0.38) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8314548 0.81 NPC1 (0.35) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed