SCHEMBL8317509

SCHEMBL8317509

COc1ccc(-c2nc3c(s2)NCCCC3)c(OC)c1OC

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 1/20 0.35
ADORA1 P30542 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
PTGS2 P35354 2/20 0.34
KDM4E B2RXH2 4/20 0.33
ALDH1A1 P00352 4/20 0.33
HPGD P15428 3/20 0.33
HSD17B10 Q99714 2/20 0.33
CRBN Q96SW2 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8315810 0.81 CYP1A1 (0.45) KDM4EALDH1A1HPGDMAPTMAPK1
Hydrochloric Acid SCHEMBL8314842 0.79 KDM4E (0.44) PTGS2KDM4EALDH1A1HPGDHSD17B10
Hydrochloric Acid SCHEMBL8315136 0.77 ACHE (0.36) KDM4EALDH1A1HPGDHSD17B10MAPT
Hydrochloric Acid SCHEMBL8315182 0.76 PARP1 (0.37) KDM4EALDH1A1HPGDHSD17B10TDP1
Hydrochloric Acid SCHEMBL8312117 0.73 RAB9A (0.42) ADORA1KDM4EALDH1A1HSD17B10TDP1
SCHEMBL10434591 0.72 PDCD1 (0.34) KDM4EALDH1A1HPGDLMNAMAPT
Oxalic Acid SCHEMBL8313128 0.72 CYP1A1 (0.40) KDM4EALDH1A1LMNAMAPTMAPK1
Oxalic Acid SCHEMBL8313123 0.72 CYP1A1 (0.40) KDM4EALDH1A1LMNAMAPTMAPK1
SCHEMBL8316374 0.72 MAPT (0.49) ADORA1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8316269 0.72 ACHE (0.39) KDM4EALDH1A1MGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0351856-B1 Thiazolo[5,4-b]azepine compounds TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-09-15 EP disclosed
US-5118806-A Enzyme inhibitor for lipoxygenase; useful for treating cancer, hepatic diseases, inflammation, cerebrovascular diseases TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-06-02 US disclosed
US-4956360-A LIPOPEROXIDE INHIBITORS, ENZYME INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-09-11 US disclosed