SCHEMBL10434591

SCHEMBL10434591

Cc1c(N)ccc(-c2nc3c(s2)NCCCC3)c1C

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 6/20 0.34
CD274 Q9NZQ7 6/20 0.34
NUDT1 P36639 1/20 0.30
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8317403 0.84 ACHE (0.39) KDM4ENPC1ALDH1A1LMNAGLA
SCHEMBL8316269 0.81 ACHE (0.39) KDM4EALDH1A1GAARAB9A
Hydrochloric Acid SCHEMBL8313444 0.79 ALDH1A1 (0.39) KDM4ENPC1ALDH1A1MAPTHPGD
Hydrochloric Acid SCHEMBL8313470 0.78 ACHE (0.40) PDCD1CD274NUDT1KDM4EALDH1A1
SCHEMBL8314378 0.77 RAB9A (0.40) KDM4ENPC1ALDH1A1LMNAMAPT
Hydrochloric Acid SCHEMBL8315904 0.76 ACHE (0.39) NUDT1KDM4EALDH1A1LMNAHPGD
Hydrochloric Acid SCHEMBL8311899 0.76 RAB9A (0.39) KDM4ENPC1ALDH1A1LMNAMAPT
SCHEMBL8314532 0.74 RAB9A (0.40) NUDT1KDM4ENPC1ALDH1A1LMNA
SCHEMBL8315862 0.74 ALOX5 (0.44) KDM4ENPC1ALDH1A1LMNAGAA
Hydrochloric Acid SCHEMBL8315136 0.74 ACHE (0.36) KDM4EALDH1A1GLAGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4956360-A LIPOPEROXIDE INHIBITORS, ENZYME INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-09-11 US claimed
EP-0351856-A2 Thiazolo[5,4-b]azepine compounds Takeda Chemical Industries, Ltd. (JP) 1990-01-24 EP claimed