SCHEMBL8318233

SCHEMBL8318233

CS(=O)(=O)c1ncc2ncnc(Nc3ccc(Cl)c([N+](=O)[O-])c3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.47
ARNT P27540 1/20 0.43
EPAS1 Q99814 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.42
BRD4 O60885 1/20 0.42
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
ERBB2 P04626 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA13 Q8N1Q1 1/20 0.40
LMNA P02545 2/20 0.39
MAPT P10636 2/20 0.39
TRPV1 Q8NER1 1/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319085 0.88 EGFR (0.44) EGFRABCG2CA1CA2CA7
SCHEMBL8317145 0.86 EGFR (0.49) EGFRERBB2HPGDHTTMAPT
SCHEMBL8318382 0.83 EGFR (0.47) EGFRARNTEPAS1ABCG2BRD4
SCHEMBL6994362 0.82 ABCG2 (0.56) EGFRABCG2
SCHEMBL6990190 0.81 EGFR (0.59) EGFRERBB2HPGDHTTMAPT
SCHEMBL8315330 0.79 EGFR (0.57) EGFRERBB2HPGDLMNAMAPT
SCHEMBL6992072 0.78 EGFR (0.44) EGFRERBB2HPGDHTTMAPT
SCHEMBL6997375 0.78 EGFR (0.47) EGFRERBB2HPGDHTTMAPT
SCHEMBL6992428 0.77 GSK3A (0.55) EGFRABCG2BRD4ERBB2HPGD
SCHEMBL6992432 0.77 GSK3A (0.55) EGFRABCG2BRD4ERBB2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed