SCHEMBL8318685

SCHEMBL8318685

O=C(NC1CC2CC3CC(C1)N2CC3=O)c1cc(Cl)cc2c1O[C@@H]1CCCC[C@@H]21

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 3/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HPGD P15428 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMYD3 Q9H7B4 2/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318689 1.00 HTR3A (0.34) HTR3ACNR1CNR2SMN1; SMN2HPGD
SCHEMBL8318695 1.00 HTR3A (0.34) HTR3ACNR1CNR2SMN1; SMN2HPGD
SCHEMBL9705653 0.83 HTR3A (0.34) HTR3A
SCHEMBL9705660 0.83 HTR3A (0.34) HTR3A
SCHEMBL9705630 0.83 HTR3A (0.34) HTR3A
SCHEMBL9706213 0.78 HTR3A (0.33) HTR3ASMYD3
SCHEMBL9678634 0.74 PTGS1 (0.38) HTR3A
SCHEMBL9678627 0.74 PTGS1 (0.38) HTR3A
SCHEMBL8323720 0.74 MEN1 (0.32)
SCHEMBL7629711 0.74 FFAR4 (0.39) HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0518767-A2 Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS INC. (US) 1992-12-16 EP claimed
US-5955470-A Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS, INC. (US) 1999-09-21 US disclosed
EP-0518767-A2 Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS INC. (US) 1992-12-16 EP disclosed