SCHEMBL8319102

SCHEMBL8319102

COC1CCC(Nc2ncc3ncnc(Nc4cccc(C)c4)c3n2)CC1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.64
ERBB2 P04626 1/20 0.51
HPGD P15428 1/20 0.51
HTT P42858 1/20 0.51
BRAF P15056 1/20 0.47
SYK P43405 1/20 0.44
KCNH2 Q12809 1/20 0.44
CSNK2A1 P68400 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319095 1.00 EGFR (0.64) EGFRERBB2HPGDHTTBRAF
SCHEMBL8319428 0.93 EGFR (0.73) EGFRERBB2HPGDHTTBRAF
SCHEMBL8314968 0.90 EGFR (0.65) EGFRERBB2HPGDHTT
SCHEMBL8314964 0.90 EGFR (0.65) EGFRERBB2HPGDHTT
SCHEMBL8319173 0.90 EGFR (0.57) EGFRERBB2HPGDHTTBRAF
SCHEMBL8319178 0.90 EGFR (0.57) EGFRERBB2HPGDHTTBRAF
SCHEMBL8318072 0.89 EGFR (0.71) EGFRERBB2HPGDHTTBRAF
SCHEMBL8318282 0.89 EGFR (0.71) EGFRERBB2HPGDHTTBRAF
SCHEMBL8313624 0.88 EGFR (0.67) EGFRERBB2HPGDHTTBRAF
SCHEMBL8319114 0.88 EGFR (0.67) EGFRERBB2HPGDHTTBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed