SCHEMBL8319299

SCHEMBL8319299

COc1ccc(N=Cc2ccc(O)c(OC)c2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.69
PTGS1 P23219 3/20 0.69
NFE2L2 Q16236 1/20 0.65
S100B P04271 1/20 0.65
BRAF P15056 1/20 0.59
ALOX5 P09917 1/20 0.55
CA12 O43570 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
CXCL12 P48061 1/20 0.53
MAPT P10636 2/20 0.53
GAA P10253 1/20 0.53
ALDH1A1 P00352 2/20 0.53
HPGD P15428 2/20 0.53
TRPA1 O75762 1/20 0.53
TRIM24 O15164 1/20 0.53
ALDH5A1 P51649 1/20 0.53
ABAT P80404 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
TRIM33 Q9UPN9 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319294 1.00 PTGS2 (0.69) PTGS2PTGS1NFE2L2S100BBRAF
SCHEMBL28507952 0.88 PTGS2 (0.69) PTGS2PTGS1CXCL12MAPTALDH1A1
SCHEMBL29351511 0.88 S100B (0.69) PTGS2PTGS1S100BALOX5CA12
SCHEMBL8325328 0.86 S100B (0.66) PTGS2PTGS1NFE2L2S100BCA12
SCHEMBL28607191 0.86 PTGS2 (0.65) PTGS2PTGS1S100BCA12CA2
SCHEMBL8325327 0.86 S100B (0.66) PTGS2PTGS1NFE2L2S100BCA12
SCHEMBL31318312 0.85 PTGS2 (0.66) PTGS2PTGS1NFE2L2MAPTALDH1A1
SCHEMBL10486517 0.84 PTGS2 (0.64) PTGS2PTGS1MAPTGAAALDH1A1
SCHEMBL10486520 0.84 PTGS2 (0.64) PTGS2PTGS1MAPTGAAALDH1A1
SCHEMBL16885013 0.84 PTGS2 (0.64) PTGS2PTGS1NFE2L2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990137-A ANTIINFLAMMATION AGENTS; PREVENTING THE OXIDATING BURST FROM PHAGOCYTIC LEUKOCYTES; CONTROLLING FREE RADICALS IN THE IMMUNE RESPONSE IDUN PHARMACEUTICALS, INC. (US) 1999-11-23 US disclosed
US-5939460-A Method of inhibiting NADPH oxidase IDUN PHARMACEUTICALS, INC. (US) 1999-08-17 US disclosed
WO-1998001120-A1 METHOD OF INHIBITING NADPH OXIDASE IDUN PHARMACEUTICALS, INCORPORATED (US) 1998-01-15 WO disclosed