SCHEMBL8320448

SCHEMBL8320448

O=c1c2sc3nsnc3sc=2c(=O)n1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.47
GSK3B P49841 7/20 0.44
GSK3A P49840 5/20 0.44
GAA P10253 2/20 0.39
KAT2B Q92831 1/20 0.36
POLB P06746 2/20 0.36
HPGD P15428 2/20 0.36
ALDH1A1 P00352 2/20 0.36
PDE1B Q01064 1/20 0.36
PDE3A Q14432 1/20 0.36
PDE11A Q9HCR9 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP2C9 P11712 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306506 0.72 MAPK1 (0.71) MAPK1GSK3BGSK3AGAAPOLB
SCHEMBL1730607 0.71 MAPK1 (0.58) MAPK1GSK3BGSK3AGAAHPGD
SCHEMBL10438652 0.69 MAPK1 (0.60) MAPK1GSK3BGSK3AGAAPOLB
SCHEMBL12660977 0.68 MAPK1 (0.65) MAPK1GSK3BGSK3AGAAKAT2B
SCHEMBL26558990 0.66 MAPK1 (0.62) MAPK1GSK3BGSK3AGAAKAT2B
SCHEMBL8208644 0.66 MAPK1 (0.56) MAPK1GSK3BGSK3AGAAPOLB
SCHEMBL13310390 0.65 MAPK1 (0.74) MAPK1GSK3BGSK3AGAAPOLB
SCHEMBL10607179 0.63 MAPK1 (0.71) MAPK1GSK3BGSK3AGAAPOLB
SCHEMBL12211923 0.63 MAPK1 (0.52) MAPK1GSK3BGSK3AGAAPOLB
SCHEMBL1722780 0.62 GSK3B (0.71) MAPK1GSK3BGSK3AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912580-A2 5H-PYRROLO(3',4':5,6)(1,4)DITHIINO(2,3-C)-(1,2,5)THIADIAZOLE-5,7(6H)-DIONE, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1999-05-06 EP claimed
WO-1998001452-A2 5H-PYRROLO(3',4':5,6)(1,4)DITHIINO(2,3-C)-(1,2,5)THIADIAZOLE-5,7(6H)-DIONE, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1998-01-15 WO claimed
US-5633219-A 5H-pyrrolo(3',4':5,6)(1,4)dithiino(2,3-C)(1,2,5)thiadiazole-5,7(6H)-dione, compositions containing them and their use as antimicrobial and marine antifouling agents THE DOW CHEMICAL COMPANY (US) 1997-05-27 US claimed
US-5633219-A 5H-pyrrolo(3',4':5,6)(1,4)dithiino(2,3-C)(1,2,5)thiadiazole-5,7(6H)-dione, compositions containing them and their use as antimicrobial and marine antifouling agents THE DOW CHEMICAL COMPANY (US) 1997-05-27 US disclosed