SCHEMBL8322126

SCHEMBL8322126

COc1ccc(C2CCN(C(C)=O)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QDPR P09417 2/20 0.63
HSD11B1 P28845 1/20 0.58
DRD2 P14416 1/20 0.55
ALDH1A1 P00352 4/20 0.53
LMNA P02545 2/20 0.53
RAB9A P51151 1/20 0.53
DRD3 P35462 1/20 0.51
MAPT P10636 2/20 0.51
FAAH O00519 1/20 0.51
BACE1 P56817 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
PDE4B Q07343 1/20 0.49
HPGD P15428 2/20 0.49
HIF1A Q16665 1/20 0.49
POLB P06746 1/20 0.49
GAA P10253 1/20 0.49
CHRM4 P08173 1/20 0.48
MTNR1B P49286 1/20 0.48
KDM4E B2RXH2 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20805979 0.91 ALDH1A1 (0.61) QDPRHSD11B1DRD2ALDH1A1LMNA
SCHEMBL2636579 0.87 HSD11B1 (0.61) QDPRHSD11B1DRD2ALDH1A1LMNA
SCHEMBL7284775 0.86 QDPR (0.57) QDPRHSD11B1ALDH1A1LMNAMAPT
SCHEMBL14412855 0.86 HSD11B1 (0.56) QDPRHSD11B1DRD2ALDH1A1LMNA
SCHEMBL23397304 0.83 ALDH1A1 (0.51) HSD11B1ALDH1A1LMNARAB9ADRD3
SCHEMBL21051331 0.83 ALDH1A1 (0.66) HSD11B1ALDH1A1LMNARAB9AMAPT
SCHEMBL14590572 0.82 QDPR (0.61) QDPRHSD11B1DRD2ALDH1A1LMNA
SCHEMBL25174711 0.82 HSD11B1 (0.70) HSD11B1DRD2ALDH1A1LMNARAB9A
SCHEMBL19066022 0.82 ALDH1A1 (0.55) QDPRHSD11B1DRD2ALDH1A1LMNA
SCHEMBL7277302 0.81 QDPR (0.69) QDPRALDH1A1POLBKDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018054549-A1 6-MEMBERED CYCLIC AMINES OR LACTAMES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2018-03-29 WO disclosed
EP-1592426-B1 2-CYANOPYRROLOPYRIMIDINES AND PHARMACEUTICAL USES THEREOF NOVARTIS AG (CH) 2007-12-19 EP disclosed
WO-2004069256-A1 2-CYANOPYRROLOPYRIMIDINES AND PHARMACEUTICAL USES THEREOF NOVARTIS AG (CH) 2004-08-19 WO disclosed