SCHEMBL8322673

SCHEMBL8322673

CC(C)(C)c1ccc(-n2nc3c(ncc4ccccc43)c2O)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 3/20 0.36
PMM2 O15305 1/20 0.34
MPI P34949 1/20 0.34
PHOSPHO1 Q8TCT1 1/20 0.34
LMNA P02545 4/20 0.34
TP53 P04637 1/20 0.34
HSD17B2 P37059 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
LHCGR P22888 1/20 0.33
UQCRB P14927 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
PLA2G10 O15496 1/20 0.33
KDM4E B2RXH2 1/20 0.33
FABP3 P05413 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324694 0.87 MAPT (0.40) MPIPHOSPHO1TRPV1KDM4ERAB9A
SCHEMBL8321754 0.85 KDM4E (0.41) SMN1; SMN2LMNATP53POLBGAA
SCHEMBL8466029 0.85 SCN9A (0.32) SMN1; SMN2MEN1KMT2ANPC1LMNA
SCHEMBL8322376 0.83 SMN1; SMN2 (0.49) SMN1; SMN2KMT2ANPC1LMNAGAA
SCHEMBL8462048 0.83 KDM4E (0.39) SMN1; SMN2MEN1KMT2ANPC1LMNA
SCHEMBL8320446 0.83 NPC1 (0.49) SMN1; SMN2MEN1KMT2ANPC1LMNA
SCHEMBL8329043 0.79 TEAD1 (0.39) SMN1; SMN2TP53TRPM8
SCHEMBL8466300 0.77 GAA (0.43) SMN1; SMN2NPC1LMNATP53POLB
SCHEMBL8329140 0.77 KMT2A (0.47) SMN1; SMN2MEN1KMT2ANPC1LMNA
Water SCHEMBL8462183 0.76 SMN1; SMN2 (0.36) AURKASMN1; SMN2MEN1KMT2APMM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888347-A1 PHARMACEUTICALLY USEFUL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-01-07 EP claimed
WO-1997034893-A1 PHARMACEUTICALLY USEFUL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-09-25 WO claimed
EP-0888347-A1 PHARMACEUTICALLY USEFUL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-01-07 EP disclosed
WO-1997034893-A1 PHARMACEUTICALLY USEFUL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-09-25 WO disclosed