SCHEMBL8322828

SCHEMBL8322828

CCOC(=O)c1cc(N)c(C)nc1C(=O)OCC

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.51
ALDH1A1 P00352 6/20 0.50
HSD17B10 Q99714 4/20 0.50
CYP1A2 P05177 1/20 0.50
TSHR P16473 3/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
GAA P10253 3/20 0.45
MAPK1 P28482 1/20 0.45
ALOX15 P16050 3/20 0.44
HSP90AA1 P07900 1/20 0.44
MAPT P10636 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 1/20 0.43
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318983 0.87 ALDH1A1 (0.50) KDM4EALDH1A1HSD17B10CYP1A2TSHR
SCHEMBL13285824 0.84 KDM4E (0.51) KDM4EALDH1A1HSD17B10TSHRMEN1
SCHEMBL9800425 0.83 KDM4E (0.50) KDM4EALDH1A1HSD17B10CYP1A2TSHR
SCHEMBL8661094 0.81 ALDH1A1 (0.50) KDM4EALDH1A1HSD17B10CYP1A2TSHR
SCHEMBL9315414 0.81 SMN1; SMN2 (0.56) KDM4EALDH1A1HSD17B10CYP1A2TSHR
SCHEMBL8319338 0.80 KDM4E (0.46) KDM4EALDH1A1HSD17B10TSHRGAA
SCHEMBL9205477 0.79 TSHR (0.49) KDM4EALDH1A1HSD17B10CYP1A2TSHR
SCHEMBL27140789 0.79 KDM4E (0.67) KDM4EALDH1A1HSD17B10TSHRMEN1
SCHEMBL31607744 0.79 KDM4E (0.67) KDM4EALDH1A1HSD17B10TSHRMEN1
SCHEMBL7471868 0.79 ALDH1A1 (0.63) KDM4EALDH1A1HSD17B10CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5959116-A 5-NITRO PYRIDINE-2,3-DICARBOXYLIC ACID ESTER CHEMICAL INTERMEDIATES MADE BY REACTING THE N-OXIDES OF PYRIDINE-2,3-DICARBOXYLIC ACID ESTERS WITH NITRIC ACID OR SODIUM NITRATE, THEN REMOVING THE N-OXIDE GROUP BASF AKTIENGESELLSCHAFT (DE) 1999-09-28 US disclosed
US-5840904-A Fluoro-pyridine-2,3-dicarboxylic anhydrides which are intermediates for herbicidal pyridine-2,3-dicarboximides BASF AKTIENGESELLSCHAFT (DE) 1998-11-24 US disclosed
US-5679622-A HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1997-10-21 US disclosed
US-5571774-A HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1996-11-05 US disclosed