SCHEMBL8322927

SCHEMBL8322927

[CH2]CC(N)(c1ccccc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.49
TSHR P16473 2/20 0.47
MAPK1 P28482 1/20 0.47
ALDH1A1 P00352 1/20 0.46
IDO1 P14902 4/20 0.46
TDO2 P48775 2/20 0.46
PNMT P11086 1/20 0.45
TAAR1 Q96RJ0 1/20 0.44
TACR1 P25103 1/20 0.43
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
ACP3 P15309 2/20 0.41
SLC6A4 P31645 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
IDH2 P48735 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8321366 0.86 ALDH1A1 (0.58) KIF11TSHRALDH1A1IDO1TDO2
SCHEMBL8322782 0.86 ALDH1A1 (0.58) KIF11TSHRALDH1A1IDO1TDO2
SCHEMBL27525548 0.82 KCNN4 (0.52) KIF11TSHRALDH1A1TAAR1HTT
SCHEMBL8321948 0.81 KIF11 (0.49) KIF11IDO1TDO2TAAR1APP
SCHEMBL8321573 0.81 KIF11 (0.49) KIF11IDO1TDO2TAAR1APP
SCHEMBL8323195 0.79 TSHR (0.48) TSHRMAPK1ALDH1A1MEN1KMT2A
SCHEMBL8324380 0.78 KIF11 (0.50) KIF11TSHRTAAR1
SCHEMBL8324065 0.78 KIF11 (0.50) KIF11ALDH1A1PNMTTAAR1
Benzene SCHEMBL8568955 0.77 TSHR (0.67) KIF11TSHRMAPK1ALDH1A1IDO1
SCHEMBL8324979 0.76 TSHR (0.45) KIF11TSHRMAPK1ALDH1A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed