SCHEMBL8323648

SCHEMBL8323648

CCOC(=O)C1=C(c2ccc(-n3c(C)nc4ncccc43)cc2)NC(C)=C(C(=O)O)C1C(C)C

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 11/20 0.45
TMIGD3 P0DMS9 2/20 0.38
TRPV1 Q8NER1 3/20 0.37
KDM4E B2RXH2 2/20 0.37
CASP1 P29466 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
ADORA2A P29274 2/20 0.35
ADORA2B P29275 2/20 0.35
TSHR P16473 1/20 0.35
CYP3A4 P08684 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328228 0.85 ADORA3 (0.44) ADORA3TMIGD3TRPV1KDM4ECASP1
SCHEMBL8523478 0.83 ADORA3 (0.43) ADORA3
SCHEMBL8327956 0.80 ADORA3 (0.49) ADORA3TMIGD3TRPV1KDM4ECASP1
SCHEMBL7873236 0.73 ADORA3 (0.40) ADORA3TMIGD3TRPV1HSD17B10ALDH1A1
SCHEMBL7873250 0.73 ADORA3 (0.37) ADORA3TMIGD3TRPV1ALDH1A1TSHR
SCHEMBL8523663 0.72 ADORA3 (0.42) ADORA3TRPV1
SCHEMBL8326446 0.70 ADORA3 (0.46) ADORA3TRPV1SIRT2SIRT1
SCHEMBL8326915 0.69 ADORA3 (0.41) ADORA3TMIGD3
SCHEMBL8323291 0.69 ADORA3 (0.43) ADORA3TRPV1
SCHEMBL8325678 0.69 ADORA3 (0.42) ADORA3TMIGD3TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0943615-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 1999-09-22 EP disclosed