Pivalamide

Pivalamide

SCHEMBL8323779

CC(C)(C)C(N)=O.NC1CCCC1c1ccc(F)cc1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.46
NR3C2 P08235 1/20 0.42
SLC9A1 P19634 1/20 0.41
HRH3 Q9Y5N1 1/20 0.39
SLC6A3 Q01959 5/20 0.38
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
KCNN4 O15554 1/20 0.38
RPS6KB1 P23443 2/20 0.36
SIGMAR1 Q99720 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17864289 0.84 KDM1A (0.63) KDM1ANR3C2SLC9A1HRH3SLC6A3
SCHEMBL3717972 0.84 KDM1A (0.63) KDM1ANR3C2SLC9A1HRH3SLC6A3
SCHEMBL4260027 0.84 KDM1A (0.63) KDM1ANR3C2SLC9A1HRH3SLC6A3
SCHEMBL1645757 0.84 KDM1A (0.63) KDM1ANR3C2SLC9A1HRH3SLC6A3
SCHEMBL7898071 0.84 KDM1A (0.63) KDM1ANR3C2SLC9A1HRH3SLC6A3
SCHEMBL3717970 0.84 KDM1A (0.63) KDM1ANR3C2SLC9A1HRH3SLC6A3
SCHEMBL13598557 0.81 KDM1A (0.63) KDM1ANR3C2SLC9A1SLC6A3SLC6A2
SCHEMBL4608144 0.73 SLC9A1 (0.50) KDM1ANR3C2SLC9A1HRH3SLC6A3
SCHEMBL1644777 0.73 SLC6A2 (0.48) KDM1ASLC6A3SLC6A2SLC6A4
SCHEMBL27992795 0.70 RPS6KB1 (0.41) KDM1AHRH3SLC6A3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858444-A4 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1999-12-01 EP disclosed
EP-0858444-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-08-19 EP disclosed
WO-1997014671-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-04-24 WO disclosed