SCHEMBL8324461

SCHEMBL8324461

OC[C@@H]1CCn2c(cc3ccccc32)C1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.48
HTR2C P28335 5/20 0.48
SIGMAR1 Q99720 9/20 0.45
PRKCE Q02156 2/20 0.39
MYLK Q15746 2/20 0.39
PRKCB P05771 2/20 0.38
HTR1A P08908 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318760 1.00 HTR2A (0.48) HTR2AHTR2CSIGMAR1PRKCEMYLK
SCHEMBL1991214 1.00 HTR2A (0.48) HTR2AHTR2CSIGMAR1PRKCEMYLK
SCHEMBL8657682 0.91 HTR2A (0.46) HTR2AHTR2CSIGMAR1
SCHEMBL8654361 0.87 HTR2A (0.54) HTR2AHTR2CSIGMAR1HTR1A
SCHEMBL8655904 0.85 PRKCE (0.51) HTR2AHTR2CSIGMAR1PRKCEMYLK
SCHEMBL8653081 0.84 HTR2A (0.43) HTR2AHTR2CSIGMAR1PRKCB
SCHEMBL8449854 0.83 SIGMAR1 (0.49) HTR2AHTR2CSIGMAR1PRKCEMYLK
SCHEMBL8451901 0.81 HTR2A (0.42) HTR2AHTR2CSIGMAR1PRKCEMYLK
SCHEMBL1993818 0.81 HTR2A (0.45) HTR2AHTR2CSIGMAR1PRKCEMYLK
SCHEMBL8451898 0.81 HTR2A (0.42) HTR2AHTR2CSIGMAR1PRKCEMYLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574783-B1 Asymmetric hydrogenation HOFFMANN LA ROCHE (CH) 1999-10-06 EP disclosed
US-5374727-A Using rhodium-diphosphine complex as hydrogenation catalyst HOFFMANN-LA ROCHE INC. (US) 1994-12-20 US disclosed
EP-0574783-A2 Asymmetric hydrogenation F. HOFFMANN-LA ROCHE AG (CH) 1993-12-22 EP disclosed