SCHEMBL8324686

SCHEMBL8324686

CCOC(=O)c1cc2cc(O[Si](C)(C)C(C)(C)C)ccc2o1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.54
CA9 Q16790 5/20 0.54
CA1 P00915 4/20 0.54
MAOB P27338 2/20 0.49
PIM1 P11309 1/20 0.45
FLT3 P36888 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CA2 P00918 1/20 0.44
CA3 P07451 1/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1390713 0.83 CA12 (0.60) CA12CA9CA1PIM1FLT3
SCHEMBL7795617 0.83 PIM1 (0.60) CA12CA9CA1PIM1FLT3
SCHEMBL8118515 0.82 MAOB (0.55) CA12CA9MAOBPIM1FLT3
SCHEMBL648621 0.82 MAOB (0.70) CA12CA9MAOBKDM4EALDH1A1
SCHEMBL6867907 0.81 MAOB (0.54) CA12CA9MAOBFLT3KDM4E
SCHEMBL31474440 0.80 ALDH1A1 (0.67) KDM4EMEN1ALDH1A1MAPTHPGD
SCHEMBL26882627 0.80 ALDH1A1 (0.67) KDM4EMEN1ALDH1A1MAPTHPGD
SCHEMBL8328098 0.79 CA12 (0.50) CA12CA9CA1MAOBALDH1A1
SCHEMBL18591911 0.79 MAOB (0.52) CA12CA9CA1MAOBFLT3
SCHEMBL18611964 0.79 MAOB (0.52) CA12CA9CA1MAOBFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed