SCHEMBL8324809

SCHEMBL8324809

COc1nc(C(Cc2cccc(Br)c2)OCc2ccccc2)ccc1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PARP15 Q460N3 1/20 0.39
CTSS P25774 7/20 0.38
CTSB P07858 6/20 0.38
BACE1 P56817 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
MCL1 Q07820 1/20 0.36
BAK1 Q16611 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CTSL P07711 5/20 0.36
CTSK P43235 3/20 0.36
KDM5A P29375 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
LRRK2 Q5S007 1/20 0.35
FFAR1 O14842 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326041 0.92 PDCD1 (0.40) PARP15CTSSCTSBBACE1MAOA
SCHEMBL8323811 0.82 CTSS (0.39) CTSSCTSBMAOAMAOBCTSL
SCHEMBL8321888 0.80 PARP15 (0.42) PARP15CTSSCTSBCTSLCTSK
SCHEMBL8324996 0.76 CTSS (0.43) PARP15CTSSCTSBMAOBCTSL
SCHEMBL8321376 0.75 MAOB (0.45) TDP1CTSSCTSBMAOAMAOB
SCHEMBL8327208 0.74 MMP1 (0.39) PARP15CTSSCTSBMAOAMAOB
SCHEMBL8325139 0.73 PARP15 (0.45) POLBPARP15CTSSCTSBMAOA
SCHEMBL8326543 0.73 LRRK2 (0.36) CTSSCTSBCTSLCTSKLRRK2
SCHEMBL8322939 0.72 MAOB (0.44) PARP15CTSSCTSBMAOAMAOB
SCHEMBL8326572 0.71 MEN1 (0.38) CTSSCTSBMAOAMAOBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed