SCHEMBL8326543

SCHEMBL8326543

O=C(Nc1nnn[nH]1)c1ccc(C(Cc2cccc(Br)c2)OCc2ccccc2)nc1Cl

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 8/20 0.36
CTSS P25774 6/20 0.34
CTSB P07858 5/20 0.34
CTSL P07711 4/20 0.34
CTSK P43235 2/20 0.34
MET P08581 1/20 0.33
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323811 0.81 CTSS (0.39) CTSSCTSBCTSLCTSK
SCHEMBL8321888 0.81 PARP15 (0.42) CTSSCTSBCTSLCTSK
SCHEMBL8326541 0.74 LRRK2 (0.47) LRRK2
SCHEMBL8324809 0.73 POLB (0.39) LRRK2CTSSCTSBCTSLCTSK
SCHEMBL8326041 0.72 PDCD1 (0.40) LRRK2CTSSCTSBCTSLCTSK
SCHEMBL8321008 0.67 GABRG2 (0.35) CTSSCTSBCTSLCTSK
SCHEMBL11561500 0.67 LRRK2 (0.63) LRRK2
SCHEMBL11560468 0.67 MET (0.52) LRRK2MET
SCHEMBL8324996 0.66 CTSS (0.43) CTSSCTSBCTSLCTSKGLA
SCHEMBL8675246 0.65 LRRK2 (0.44) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed