SCHEMBL8324826

SCHEMBL8324826

COCN1C(=O)N(Cc2ccccc2)N=C(c2ccc(Cl)cc2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 1/20 0.46
TP53 P04637 2/20 0.41
CES1 P23141 2/20 0.41
CES2 O00748 1/20 0.41
BCHE P06276 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
PRKAG1 P54619 1/20 0.40
PRKAA2 P54646 1/20 0.40
PRKAB1 Q9Y478 1/20 0.40
CCKBR P32239 2/20 0.40
NPSR1 Q6W5P4 2/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
ALDH1A1 P00352 2/20 0.38
ALDH2 P05091 2/20 0.38
ALDH3A1 P30838 2/20 0.38
CHRM1 P11229 1/20 0.38
UTS2R Q9UKP6 1/20 0.37
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9705380 0.78 PTH1R (0.50) PTH1RTP53CES1CES2BCHE
SCHEMBL8322539 0.76 TP53 (0.42) TP53CES1CES2BCHEPTGDR2
SCHEMBL8315954 0.72 CCKBR (0.43) PTH1RCCKBRNPSR1HTTALDH1A1
SCHEMBL8317832 0.71 BRD4 (0.55) CCKBR
SCHEMBL8318719 0.69 BRD4 (0.49) CCKBR
SCHEMBL9703671 0.68 PTH1R (0.49) PTH1RCCKBRNPSR1GAAHTT
SCHEMBL8315258 0.68 BRD4 (0.46)
SCHEMBL9703395 0.68 PGR (0.53) PTH1RTP53CES1BCHECCKBR
SCHEMBL8318456 0.68 BRD4 (0.55) CCKBR
SCHEMBL8316213 0.67 BRD4 (0.55) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934940-A1 CYTOKINE PRODUCTION INHIBITORS, TRIAZEPINE COMPOUNDS, AND INTERMEDIATES THEREOF Japan Tobacco Inc. (JP) 1999-08-11 EP disclosed
EP-0792880-A1 OSTEOPOROSIS REMEDY AND TRIAZEPINE COMPOUND Japan Tobacco Inc. (JP) 1997-09-03 EP disclosed