SCHEMBL8324850

SCHEMBL8324850

CCCOC(=O)c1c(NC2CN(Cc3ccc(C(F)(F)F)cc3)CCO2)n(-c2ccccc2)c(=S)n(C)c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 6/20 0.38
FAAH O00519 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
GAA P10253 1/20 0.35
CYP2C19 P33261 1/20 0.35
DRD2 P14416 3/20 0.34
DRD3 P35462 2/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
SIGMAR1 Q99720 3/20 0.34
TEAD1 P28347 1/20 0.34
HIF1A Q16665 2/20 0.33
EPAS1 Q99814 2/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
BACE1 P56817 1/20 0.33
KCNH2 Q12809 1/20 0.33
MOGAT2 Q3SYC2 1/20 0.33
OPRL1 P41146 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327984 0.92 DRD4 (0.39) DRD4CYP1A2CYP3A4GAACYP2C19
SCHEMBL8325449 0.92 DRD4 (0.42) DRD4FAAHDRD2DRD3CHRM2
SCHEMBL8323147 0.90 DRD4 (0.39) DRD4FAAHSIGMAR1
SCHEMBL8324935 0.88 DRD4 (0.38) DRD4CYP1A2CYP3A4GAACYP2C19
SCHEMBL8327102 0.84 DRD4 (0.41) DRD4GAACYP2C19DRD2DRD3
SCHEMBL8328890 0.84 DRD4 (0.41) DRD4FAAHGAADRD2DRD3
SCHEMBL8327273 0.82 DRD4 (0.40) DRD4FAAHDRD2DRD3SIGMAR1
SCHEMBL8327988 0.81 DRD4 (0.39) DRD4CYP1A2CYP3A4GAACYP2C19
SCHEMBL8327903 0.81 DRD4 (0.42) DRD4FAAHDRD2DRD3SIGMAR1
SCHEMBL8326299 0.80 DRD4 (0.38) DRD4FAAHGAACHRM1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed