SCHEMBL8327102

SCHEMBL8327102

Cn1c(=O)c(C(=O)OCc2ccccc2)c(NC2CN(Cc3ccc(F)cc3)CCO2)n(-c2ccccc2)c1=S

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.41
ABL1 P00519 1/20 0.37
RIN1 Q13671 1/20 0.37
GAA P10253 2/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
DRD2 P14416 4/20 0.35
DRD3 P35462 4/20 0.35
TSHR P16473 2/20 0.35
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34
SIGMAR1 Q99720 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
CHRM4 P08173 1/20 0.34
GRIN2B Q13224 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328890 0.93 DRD4 (0.41) DRD4GAALMNAMAPTDRD2
SCHEMBL8327984 0.92 DRD4 (0.39) DRD4GAALMNAMAPTDRD3
SCHEMBL8327273 0.91 DRD4 (0.40) DRD4MAPTDRD2DRD3SIGMAR1
SCHEMBL8324935 0.91 DRD4 (0.38) DRD4GAALMNAMAPTDRD2
SCHEMBL8327988 0.90 DRD4 (0.39) DRD4GAALMNAMAPTDRD3
SCHEMBL8326299 0.88 DRD4 (0.38) DRD4GAALMNAMAPTMAPK8
SCHEMBL8325449 0.84 DRD4 (0.42) DRD4DRD2DRD3SIGMAR1
SCHEMBL8324850 0.84 DRD4 (0.38) DRD4GAADRD2DRD3SIGMAR1
SCHEMBL8327903 0.84 DRD4 (0.42) DRD4DRD2DRD3SIGMAR1
SCHEMBL8323147 0.83 DRD4 (0.39) DRD4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed