SCHEMBL8324980

SCHEMBL8324980

O=C(O)CC1(C(=O)O)CCn2c(cc3ccccc32)C1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.42
HTR2C P28335 5/20 0.42
SIGMAR1 Q99720 15/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329532 0.88 SIGMAR1 (0.41) HTR2AHTR2CSIGMAR1
SCHEMBL8326874 0.80 HTR2A (0.42) HTR2AHTR2CSIGMAR1
SCHEMBL8328986 0.76 HTR2A (0.42) HTR2AHTR2C
SCHEMBL3156042 0.70 HTR2A (0.46) HTR2AHTR2CSIGMAR1
SCHEMBL8328249 0.67 HTR2A (0.44) HTR2AHTR2CSIGMAR1
SCHEMBL8325900 0.67 HTR2A (0.46) HTR2AHTR2CSIGMAR1
SCHEMBL8449854 0.66 SIGMAR1 (0.49) HTR2AHTR2CSIGMAR1
SCHEMBL8330362 0.65 HTR2A (0.38) HTR2AHTR2C
SCHEMBL16579978 0.65 CYP2D6 (0.55) SIGMAR1
SCHEMBL5380065 0.65 SIGMAR1 (0.64) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed