SCHEMBL8330362

SCHEMBL8330362

CCOC(=O)CC1(C(=O)OCC)Cc2cc3ccccc3n2C1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
ALDH1A1 P00352 2/20 0.38
OPRM1 P35372 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NOD2 Q9HC29 3/20 0.36
NOD1 Q9Y239 3/20 0.36
KDM4E B2RXH2 3/20 0.36
HSD17B10 Q99714 2/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
SAE1 Q9UBE0 1/20 0.36
UBA2 Q9UBT2 1/20 0.36
PSMD14 O00487 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328986 0.89 HTR2A (0.42) HTR2AHTR2CALDH1A1OPRM1MEN1
SCHEMBL8320925 0.89 HTR2A (0.42) HTR2AHTR2CALDH1A1OPRM1MEN1
SCHEMBL3156042 0.75 HTR2A (0.46) HTR2AHTR2COPRM1HPGD
SCHEMBL8326463 0.74 ALDH1A1 (0.40) ALDH1A1OPRM1MEN1KMT2ANOD2
SCHEMBL8322854 0.73 ALDH1A1 (0.36) ALDH1A1OPRM1MEN1KMT2ANOD2
SCHEMBL8325800 0.73 ALDH1A1 (0.39) HTR2AHTR2CALDH1A1MEN1KMT2A
SCHEMBL22904560 0.72 BRD4 (0.48) OPRM1MEN1KMT2ATSHRGAA
SCHEMBL8327585 0.70 OPRM1 (0.40) ALDH1A1OPRM1MEN1KMT2ANOD2
SCHEMBL8329435 0.69 HTR2A (0.39) HTR2AHTR2CALDH1A1OPRM1MEN1
SCHEMBL8322862 0.68 MEN1 (0.36) HTR2AHTR2COPRM1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed