SCHEMBL8325499

SCHEMBL8325499

[CH2]CC(c1ccccc1)c1cccc(F)c1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.49
TDO2 P48775 1/20 0.49
CNR2 P34972 1/20 0.44
CYP19A1 P11511 1/20 0.43
SLC6A4 P31645 3/20 0.41
SLC6A2 P23975 2/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
NFE2L2 Q16236 1/20 0.39
AOC3 Q16853 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 1/20 0.39
GBA1 P04062 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430169 0.81 CYP19A1 (0.44) CNR2CYP19A1SLC6A4NFE2L2
SCHEMBL94275 0.80 HTR2A (0.52)
SCHEMBL3903476 0.80 HTR2A (0.64) IDO1TDO2CNR2CYP19A1SLC6A4
SCHEMBL23126406 0.80 IDO1 (0.49) IDO1TDO2CNR2CYP19A1SLC6A4
Ammonia Solution, Strong SCHEMBL5999540 0.78 IDO1 (0.47) IDO1TDO2CNR2CYP19A1SLC6A4
SCHEMBL23021624 0.78 SLC6A2 (0.53) IDO1TDO2CNR2CYP19A1SLC6A4
Methylamine SCHEMBL6900406 0.77 IDO1 (0.50) IDO1TDO2CNR2CYP19A1SLC6A4
SCHEMBL5999535 0.77 HRH1 (0.67) IDO1TDO2CNR2CYP19A1SLC6A4
SCHEMBL8324166 0.76 ACP3 (0.47) IDO1TDO2SLC6A4SLC6A2AOC3
SCHEMBL8322755 0.76 KIF11 (0.41) SLC6A4SLC6A2HDAC4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed