SCHEMBL8325591

SCHEMBL8325591

CNC(NCC1CCCCN1Cc1ccc(F)cc1)=C(C#N)C#N

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.40
SPHK2 Q9NRA0 1/20 0.40
SPHK1 Q9NYA1 1/20 0.40
CCR2 P41597 4/20 0.38
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7495987 0.83 KMT2A (0.35) ALDH1A1
SCHEMBL8326114 0.79 MEN1 (0.48)
SCHEMBL8327662 0.78 KDM4E (0.39) SPHK2SPHK1ALDH1A1
SCHEMBL8326334 0.78 KMT2A (0.56) ALDH1A1
SCHEMBL8325593 0.75 SPHK2 (0.41) OPRM1SPHK2SPHK1ALDH1A1
SCHEMBL8621242 0.74 SPHK2 (0.38) OPRM1SPHK2SPHK1ALDH1A1
SCHEMBL8325845 0.74 SPHK2 (0.45) SPHK2SPHK1ALDH1A1
SCHEMBL7488935 0.73 DRD3 (0.51)
SCHEMBL8328838 0.72 MAPK1 (0.50)
SCHEMBL8329414 0.72 SIGMAR1 (0.53) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
EP-0760362-A1 NOVEL DIAMINOMETHYLIDENE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed