SCHEMBL8329414

SCHEMBL8329414

CNC(NC1CCN(Cc2ccc(F)cc2)CC1)=C(C#N)C#N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.53
PRKAA2 P54646 4/20 0.51
MCHR1 Q99705 3/20 0.50
SLC6A12 P48065 1/20 0.50
TMEM97 Q5BJF2 1/20 0.50
ALDH1A1 P00352 1/20 0.48
BCHE P06276 2/20 0.48
ACHE P22303 2/20 0.48
BACE1 P56817 2/20 0.48
DRD3 P35462 1/20 0.47
CCR3 P51677 1/20 0.47
CYP2D6 P10635 1/20 0.46
CHRM1 P11229 1/20 0.46
HTR2A P28223 1/20 0.46
PRKAB2 O43741 2/20 0.46
PRKAG1 P54619 2/20 0.46
PRKAA1 Q13131 2/20 0.46
PRKAG3 Q9UGI9 2/20 0.46
PRKAG2 Q9UGJ0 2/20 0.46
PRKAB1 Q9Y478 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328601 0.89 BCHE (0.41) SIGMAR1PRKAA2MCHR1ALDH1A1BCHE
SCHEMBL8326114 0.84 MEN1 (0.48)
SCHEMBL4383023 0.80 DPP7 (0.62) SIGMAR1MCHR1SLC6A12TMEM97ALDH1A1
SCHEMBL8328838 0.79 MAPK1 (0.50) ACHE
SCHEMBL7491968 0.77 OPRK1 (0.44) DRD3CCR3
SCHEMBL8151042 0.76 BCHE (0.62) SIGMAR1PRKAA2MCHR1SLC6A12TMEM97
SCHEMBL8326334 0.76 KMT2A (0.56) MCHR1ALDH1A1BCHECCR3ATM
SCHEMBL8329774 0.75 MAPK1 (0.48)
SCHEMBL8713729 0.74 GAA (0.50) SIGMAR1PRKAA2CCR3PRKAB2PRKAG1
SCHEMBL4388051 0.73 DPP7 (0.54) SIGMAR1MCHR1SLC6A12TMEM97ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5753654-A GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-05-19 US disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760362-A1 NOVEL DIAMINOMETHYLIDENE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed