SCHEMBL8325622

SCHEMBL8325622

CC(C[CH]c1ccc(F)cc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.44
TAAR1 Q96RJ0 3/20 0.42
POLB P06746 1/20 0.41
AOC3 Q16853 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPC1 O15118 1/20 0.38
TRPA1 O75762 2/20 0.38
RIPK1 Q13546 1/20 0.38
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14910878 0.87 TAAR1 (0.50) TAAR1AOC3TRPA1RIPK1
SCHEMBL8325764 0.84 TAAR1 (0.44) TAAR1AOC3TRPA1RIPK1SMN1; SMN2
SCHEMBL8329048 0.81 NPC1 (0.46) TAAR1POLBCYP3A4CYP2D6CYP2C9
SCHEMBL8325507 0.79 TRPA1 (0.50) TAAR1TRPA1ALDH1A1
SCHEMBL8327108 0.79 NFE2L2 (0.44) NFE2L2ALDH1A1MAPTALOX15TSHR
SCHEMBL8327482 0.78 CYP3A4 (0.42) TAAR1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL19317395 0.75 TRPA1 (0.53) TAAR1POLBAOC3CYP3A4CYP2D6
SCHEMBL8326387 0.74 TAAR1 (0.41) TAAR1AOC3CYP3A4TRPA1RIPK1
SCHEMBL8324571 0.72 TP53 (0.43) TAAR1AOC3NPC1TRPA1RIPK1
SCHEMBL15515987 0.72 NFE2L2 (0.48) NFE2L2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed