SCHEMBL8329048

SCHEMBL8329048

CC(C[CH]c1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
TSHR P16473 2/20 0.41
ALDH1A1 P00352 2/20 0.41
ACP3 P15309 1/20 0.41
KIF11 P52732 1/20 0.40
SLC6A4 P31645 5/20 0.40
LMNA P02545 5/20 0.40
SLC6A2 P23975 4/20 0.40
SLC6A3 Q01959 4/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2C19 P33261 3/20 0.40
CYP3A4 P08684 3/20 0.40
HRH3 Q9Y5N1 2/20 0.40
MTOR P42345 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
MAPK1 P28482 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324977 0.83 IDO1 (0.49) NPC1RAB9AALDH1A1ACP3MEN1
SCHEMBL14910878 0.82 TAAR1 (0.50) HTR2ATAAR1RIPK1
SCHEMBL8325622 0.81 NFE2L2 (0.44) NPC1TSHRALDH1A1CYP2D6CYP2C19
SCHEMBL8322780 0.81 TACR1 (0.46) NPC1RAB9ATSHRALDH1A1ACP3
SCHEMBL8325764 0.80 TAAR1 (0.44) TSHRLMNAACHETAAR1SMN1; SMN2
SCHEMBL8325507 0.75 TRPA1 (0.50) ALDH1A1ACP3MEN1KMT2ATAAR1
SCHEMBL28724553 0.73 PDE2A (0.42) TSHRALDH1A1ACP3CYP2D6CYP2C19
SCHEMBL28724552 0.73 PDE2A (0.42) TSHRALDH1A1ACP3CYP2D6CYP2C19
SCHEMBL17071860 0.71 ACP3 (0.55) NPC1RAB9ATSHRALDH1A1ACP3
SCHEMBL8326251 0.71 NPC1 (0.59) NPC1RAB9ATSHRALDH1A1KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed