SCHEMBL8325682

SCHEMBL8325682

CCCc1c(CNc2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s2)cnc2nc(N)nc(N)c12

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GART P22102 1/20 0.49
DHFR P00374 6/20 0.46
TYMS P04818 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326393 0.89 TYMS (0.51) GARTDHFRTYMS
SCHEMBL8318241 0.86 DHFR (0.55) DHFR
SCHEMBL9067311 0.81 DHFR (0.54) DHFR
SCHEMBL9067195 0.78 DHFR (0.51) GARTDHFRTYMS
SCHEMBL9069620 0.76 DHFR (0.53) DHFRTYMS
SCHEMBL15057071 0.76 DHFR (0.59) GARTDHFRTYMS
SCHEMBL15057068 0.76 DHFR (0.59) GARTDHFRTYMS
SCHEMBL8325555 0.75 DHFR (0.54) GARTDHFRTYMS
SCHEMBL9379640 0.74 TYMS (0.56) GARTDHFRTYMS
SCHEMBL9379643 0.74 TYMS (0.56) GARTDHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0638079-B1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION STANFORD RES INST INT (US) 1999-12-15 EP disclosed
US-5536724-A Antiinflammatory and antineoplastic 5-deazaaminopterins and 5,10-dideazaaminopterins SRI INTERNATIONAL (US) 1996-07-16 US disclosed
EP-0638079-A1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION SRI INTERNATIONAL (US) 1995-02-15 EP disclosed
WO-1993022312-A1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION SRI INTERNATIONAL (US) 1993-11-11 WO disclosed