SCHEMBL8325787

SCHEMBL8325787

O=C(O)C1Cc2cc3ccccc3n2CC1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.40
HTR2C P28335 4/20 0.40
DAO P14920 1/20 0.39
SIGMAR1 Q99720 10/20 0.39
MCL1 Q07820 1/20 0.38
NOTUM Q6P988 1/20 0.38
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8449826 0.84 MAPT (0.42) HTR2AHTR2CDAOSIGMAR1MCL1
SCHEMBL8452782 0.76 HTR2A (0.44) HTR2AHTR2CSIGMAR1NOTUM
SCHEMBL8454162 0.76 HTR2A (0.44) HTR2AHTR2CSIGMAR1NOTUM
SCHEMBL8447696 0.76 HTR2A (0.43) HTR2AHTR2CDAOSIGMAR1NOTUM
SCHEMBL30684404 0.76 HTR2A (0.44) HTR2AHTR2CSIGMAR1NOTUM
SCHEMBL18229903 0.76 HTR2A (0.42) HTR2AHTR2CSIGMAR1NOTUM
SCHEMBL18229914 0.76 HTR2A (0.42) HTR2AHTR2CSIGMAR1NOTUM
SCHEMBL18229904 0.76 HTR2A (0.42) HTR2AHTR2CSIGMAR1NOTUM
SCHEMBL8448458 0.74 SIGMAR1 (0.42) HTR2AHTR2CSIGMAR1
SCHEMBL18911725 0.73 HTR2A (0.46) HTR2AHTR2CSIGMAR1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed