SCHEMBL8448458

SCHEMBL8448458

CC(C)C(=O)C1Cc2cc3ccccc3n2C1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 18/20 0.42
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8450915 0.86 HTR2A (0.43) SIGMAR1HTR2AHTR2C
SCHEMBL8446846 0.86 SIGMAR1 (0.46) SIGMAR1HTR2AHTR2C
SCHEMBL8449826 0.82 MAPT (0.42) SIGMAR1HTR2AHTR2C
SCHEMBL8447552 0.77 ALDH1A1 (0.44)
SCHEMBL8450054 0.77 HTR2A (0.48) SIGMAR1HTR2AHTR2C
SCHEMBL8453122 0.76 SIGMAR1 (0.38) SIGMAR1HTR2AHTR2C
SCHEMBL8325787 0.74 HTR2A (0.40) SIGMAR1HTR2AHTR2C
SCHEMBL18911725 0.72 HTR2A (0.46) SIGMAR1HTR2AHTR2C
SCHEMBL8454162 0.71 HTR2A (0.44) SIGMAR1HTR2AHTR2C
SCHEMBL8452782 0.71 HTR2A (0.44) SIGMAR1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0624586-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-09-01 EP disclosed
US-5721230-A ANTIINFLAMMATORY AGENT, VIRICIDES; TREATING CARDIOVASCULAR DISORDER, RESPIRATORY SYSTEM DISORDER, THROMBOSIS, DIABETES, ALOPECIA HOFFMANN-LA ROCHE INC. (US) 1998-02-24 US disclosed
EP-0624586-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1994-11-17 EP disclosed