SCHEMBL8326388

SCHEMBL8326388

[CH2]CC(C)(c1ccccc1)c1cccc(C(C)C)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.50
PTPN5 P54829 4/20 0.39
RIPK1 Q13546 1/20 0.36
HDAC4 P56524 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MDM4 O15151 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
TYR P14679 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35
CA5A P35218 1/20 0.35
HTT P42858 1/20 0.35
MDM2 Q00987 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326304 0.81 KIF11 (0.55) KIF11PTPN5HDAC4HDAC8KDM4E
SCHEMBL8463022 0.81 KIF11 (0.55) KIF11PTPN5HDAC4HDAC8KDM4E
SCHEMBL4249887 0.80 TAAR1 (0.46) ALDH1A1CYP3A4MAPTALOX15TAAR1
SCHEMBL8324574 0.77 KIF11 (0.46) KIF11PTPN5TP53CYP3A4ALOX12
SCHEMBL16191594 0.77 KIF11 (0.53) KIF11PTPN5RIPK1HDAC4HDAC8
SCHEMBL8322592 0.76 TSHR (0.46) KIF11KDM4ETP53CYP3A4MAPT
SCHEMBL8328588 0.76 KIF11 (0.45) KIF11ALDH1A1ALOX15CHRM3SCN5A
SCHEMBL8324979 0.76 TSHR (0.45) KIF11ALDH1A1TP53CYP3A4MAPT
SCHEMBL598661 0.74 KIF11 (0.49) KIF11PTPN5HDAC4HDAC8KDM4E
SCHEMBL4981920 0.74 KIF11 (0.49) KIF11PTPN5HDAC4HDAC8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed