SCHEMBL8326656

SCHEMBL8326656

CC(C)(C)OC(=O)N1CCCC2(CCn3c(cc4ccccc43)C2)C1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.48
SCD5 Q86SK9 1/20 0.44
CYP1A2 P05177 6/20 0.42
CYP3A4 P08684 5/20 0.42
CYP2C9 P11712 5/20 0.42
CYP2C19 P33261 4/20 0.42
TSHR P16473 3/20 0.42
SIGMAR1 Q99720 3/20 0.41
CYP2D6 P10635 4/20 0.40
HIF1A Q16665 1/20 0.40
HSD11B1 P28845 1/20 0.39
USP2 O75604 3/20 0.39
MAPK1 P28482 1/20 0.39
ACACB O00763 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
USP30 Q70CQ3 1/20 0.39
HDAC2 Q92769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327015 0.95 CYP11B2 (0.53) CYP11B2SCD5SIGMAR1HSD11B1ACACB
SCHEMBL8325258 0.89 CYP11B2 (0.53) CYP11B2SCD5SIGMAR1HSD11B1ACACB
SCHEMBL615033 0.76 SIGMAR1 (0.63) SIGMAR1
SCHEMBL6715677 0.74 HTR2A (0.53) SIGMAR1
SCHEMBL25164880 0.72 CYP3A4 (0.65) CYP11B2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL14240265 0.72 HPGD (0.46) CYP11B2SCD5CYP1A2CYP3A4CYP2C9
SCHEMBL25052826 0.72 HPGD (0.46) CYP11B2SCD5CYP1A2CYP3A4CYP2C9
SCHEMBL17608988 0.71 CYP2D6 (0.64) CYP1A2CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL14662248 0.71 CYP11B2 (0.42) CYP11B2SCD5CYP1A2CYP3A4CYP2C9
SCHEMBL16835523 0.70 CYP11B2 (0.40) CYP11B2SCD5CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed