SCHEMBL8327015

SCHEMBL8327015

CC(C)(C)OC(=O)N1CCC2(CCn3c(cc4ccccc43)C2)C1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.53
SCD5 Q86SK9 1/20 0.48
ACACB O00763 5/20 0.43
SIGMAR1 Q99720 1/20 0.43
USP30 Q70CQ3 2/20 0.42
HDAC2 Q92769 2/20 0.41
GPR183 P32249 1/20 0.41
SPR P35270 4/20 0.40
HDAC1 Q13547 1/20 0.39
TNKS O95271 1/20 0.39
PARP1 P09874 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
HSD11B1 P28845 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326656 0.95 CYP11B2 (0.48) CYP11B2SCD5ACACBSIGMAR1USP30
SCHEMBL8325258 0.94 CYP11B2 (0.53) CYP11B2SCD5ACACBSIGMAR1USP30
SCHEMBL615033 0.78 SIGMAR1 (0.63) SIGMAR1
SCHEMBL6715677 0.77 HTR2A (0.53) SIGMAR1CHRM2CHRM4CHRM1CHRM3
SCHEMBL14742358 0.72 SCD5 (0.64) CYP11B2SCD5ACACBUSP30TNKS
SCHEMBL8320735 0.72 SIGMAR1 (0.39) SIGMAR1USP30
SCHEMBL6868004 0.71 CYP11B2 (0.54) CYP11B2SCD5ACACBUSP30HDAC2
SCHEMBL19838586 0.71 CYP3A4 (0.66) CYP11B2SCD5USP30
SCHEMBL23902054 0.71 MAPK1 (0.51) CYP11B2SCD5CHRM2CHRM4CHRM1
SCHEMBL29609790 0.71 MAPK1 (0.51) CYP11B2SCD5CHRM2CHRM4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed