SCHEMBL8327028

SCHEMBL8327028

O=C1NCc2ccccc2C([N+](=O)[O-])N1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.36
GAA P10253 1/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
ATM Q13315 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
GPR68 Q15743 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MYC P01106 1/20 0.32
ANPEP P15144 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3416899 0.80 CYP2D6 (0.37) MEN1KMT2AMAPTALDH1A1CYP3A4
Bromide SCHEMBL10516995 0.78 CYP2D6 (0.36) MEN1KMT2AMAPTALDH1A1CYP3A4
SCHEMBL8327735 0.73 ANPEP (0.42) CA12CA9MEN1KMT2ASMN1; SMN2
SCHEMBL3824370 0.69 PRCP (0.50) GAAMEN1KMT2AMAPTALDH1A1
SCHEMBL8329852 0.67 CES1 (0.33)
SCHEMBL14061414 0.67 CA12 (0.56) GAACA12CA9
SCHEMBL4544209 0.64 TDP1 (0.45) GAATDP1MEN1KMT2AMAPT
SCHEMBL4992475 0.62 ANPEP (0.53) CA12CA9MEN1KMT2ACYP3A4
SCHEMBL22570048 0.62 CA12 (0.39) CA12CA9MEN1KMT2AMAPT
SCHEMBL14581370 0.62 CA12 (0.68) CA12CA9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed