SCHEMBL8327735

SCHEMBL8327735

NC1NC(=O)NCc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 2/20 0.42
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
HTR2A P28223 3/20 0.38
RET P07949 1/20 0.35
HTR2C P28335 1/20 0.35
HRH1 P35367 1/20 0.35
MEN1 O00255 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
MYC P01106 1/20 0.34
KDM1A O60341 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4992475 0.74 ANPEP (0.53) ANPEPCA12CA9HTR2AMEN1
SCHEMBL28816482 0.74 SMN1; SMN2 (0.54) ANPEPHTR2ARETHTR2CHRH1
SCHEMBL8327028 0.73 RAB9A (0.36) ANPEPCA12CA9MEN1CYP3A4
Bromide SCHEMBL4989971 0.73 ANPEP (0.52) ANPEPCA12CA9HTR2AMEN1
SCHEMBL27543841 0.73 HTR2A (0.48) ANPEPHTR2ARETSMN1; SMN2
Bromide SCHEMBL30630619 0.73 ANPEP (0.52) ANPEPCA12CA9HTR2AMEN1
SCHEMBL1567832 0.72 HTR2A (0.46) ANPEPHTR2AMEN1CYP3A4CYP2D6
SCHEMBL14061414 0.71 CA12 (0.56) CA12CA9
SCHEMBL7539000 0.66 IDO1 (0.43) HTR2ARETHTR2CHRH1MYC
SCHEMBL14581370 0.66 CA12 (0.68) CA12CA9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed