SCHEMBL8329852

SCHEMBL8329852

O=C1NCc2c(ccc3c2NC(=O)C3=O)C([N+](=O)[O-])N1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CES1 P23141 4/20 0.33
DAO P14920 2/20 0.33
NSD2 O96028 1/20 0.33
BCHE P06276 1/20 0.33
LIG1 P18858 1/20 0.31
CAPN9 O14815 1/20 0.31
CASP3 P42574 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329643 0.69 CES1 (0.42) CES1DAONSD2BCHELIG1
SCHEMBL8327028 0.67 RAB9A (0.36)
SCHEMBL29689350 0.61 CES1 (0.42) CES1DAONSD2BCHELIG1
SCHEMBL2973373 0.61 SMN1; SMN2 (0.47)
SCHEMBL505409 0.60 S100A4 (0.55) CES1DAONSD2BCHELIG1
SCHEMBL8329359 0.59 CES1 (0.43) CES1DAONSD2BCHELIG1
SCHEMBL8330728 0.59 CES1 (0.43) CES1DAONSD2BCHELIG1
SCHEMBL13058018 0.58 ALDH1A1 (0.50) CES1DAONSD2BCHELIG1
SCHEMBL3754645 0.58 CES1 (0.59) CES1DAONSD2BCHELIG1
SCHEMBL31355582 0.58 CES1 (0.42) CES1DAONSD2BCHELIG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed