SCHEMBL8327099

SCHEMBL8327099

CCOC(=O)CN1CCc2c(ccc3c2NC(=O)C3=O)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 2/20 0.39
PDCD1 Q15116 1/20 0.39
PIN1 Q13526 1/20 0.39
PIN4 Q9Y237 1/20 0.39
ALDH1A1 P00352 4/20 0.37
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
AOC3 Q16853 2/20 0.36
LMNA P02545 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 2/20 0.36
HSD17B10 Q99714 2/20 0.36
KDM4E B2RXH2 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330143 0.88 CD274 (0.37) CD274PDCD1PIN1PIN4ALDH1A1
SCHEMBL8330144 0.88 CD274 (0.37) CD274PDCD1PIN1PIN4ALDH1A1
SCHEMBL8328296 0.74 NOTUM (0.46) ALDH1A1LMNAMAPTHSD17B10ALOX15
SCHEMBL8326465 0.73 CES1 (0.40) KDM4ETSHRCYP2C19GSK3B
SCHEMBL8329206 0.73 CES1 (0.40) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL7399072 0.71 MAPT (0.61) ALDH1A1MEN1RAB9AKMT2ALMNA
SCHEMBL7128888 0.70 ESR1 (0.51) CD274ALDH1A1MEN1KMT2AMAPT
Hydrochloric Acid SCHEMBL8824760 0.70 MAPT (0.60) ALDH1A1MEN1RAB9AKMT2ALMNA
SCHEMBL27492242 0.69 CA9 (0.50) CD274PDCD1ALDH1A1MEN1RAB9A
SCHEMBL8325983 0.69 ESR1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed